Friday, January 18, 2013

Drug Discovery@nature.com 18 January 2013

Drug Discovery
TABLE OF CONTENTS

18 January 2013

News
Analysis
Research Highlights
Research & Reviews
Careers


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News

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Pfizer's first-in-class JAK inhibitor pricey for rheumatoid arthritis market
doi:10.1038/nbt0113-3
Pfizer's newly approved Xeljanz (tofacitinib) is poised to test the multibillion dollar rheumatoid arthritis market, currently dominated by tumor necrosis factor alpha inhibitors.
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MEK inhibitor nears approval
doi:10.1038/nbt0113-4
An FDA advisory committee has discussed materials on the MEK inhibitor trametinib, submitted by GlaxoSmithKline.
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Anthrax drug first antibacterial mAb to win approval
doi:10.1038/nbt0113-8
In mid-December, the FDA approved ABthrax, or raxibacumab, for use as an adjunct to conventional antibiotics in patients with inhalational anthrax. This approval is the first under the agency's 'animal rule'.
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Cardiac stem cell therapies inch toward clinical litmus test
doi:10.1038/nbt0113-5
Several upcoming phase 3 trials will deliver the data necessary to build a clear picture of the true potential of cell therapy in cardiac disease.
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Analysis

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mAb about FGF21
doi:10.1038/scibx.2013.1
Amgen researchers have developed an antibody that mimics fibroblast growth factor 21 and has antidiabetic effects in monkeys. The findings are informing drug development by at least six companies.
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Alzheimer's disease market: hope deferred
doi:10.1038/nrd3922
The last few months have seen a flurry of trial results for investigational agents in Alzheimer's disease. This analysis investigates the different categories of developmental drugs, and provides an outlook to the future of the market.
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Research Highlights

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Lung disorders: A new model and modulator of pulmonary oedema
doi:10.1038/nrd3917
Two complementary studies have identified a new microdevice model — termed 'lung on a chip' — of pulmonary oedema, and identified a blocker of TRPV4 that inhibits pulmonary oedema in animal models.
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Immunotherapy: Immunological bullets against Alzheimer's disease
doi:10.1038/nrd3919
The exact contribution of innate immune signalling to Alzheimer's disease pathogenesis is still unclear. Now, researchers have identified IL-12 and IL-23 signalling as a therapeutic target in this neurodegenerative disorder.
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Neurological disorders: Targeting translation in autism
doi:10.1038/nrd3915
A study in Nature shows that pharmacological inhibition of eIF4E activity or siRNA-mediated knockdown of neuroligin 1 are novel potential targets for the treatment of Autism Spectrum Disorders.
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Research & Reviews

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Objective assessment of cancer genes for drug discovery
doi:10.1038/nrd3913
This article describes and demonstrates an objective, systematic computational assessment of biological and chemical space. The approach can be applied to any human gene set to prioritize targets for further evaluation.
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Kynurenines in the CNS: recent advances and new questions
doi:10.1038/nrd3793
This Review describes the role of the kynurenine pathway in the pathology of Huntington's disease, migraine and multiple sclerosis, and highlights the most promising compounds that could be of therapeutic value.
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Ablation of TRIP-Br2, a regulator of fat lipolysis, thermogenesis and oxidative metabolism, prevents diet-induced obesity and insulin resistance
doi:10.1038/nm.3056
As expression of TRIP-Br2 is elevated in fat from obese humans, TRIP-Br2 might be a new therapeutic target against insulin resistance and hyperlipidemia.
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ABT-199, a potent and selective BCL-2 inhibitor, achieves antitumor activity while sparing platelets
doi:10.1038/nm.3048
The authors have engineered anti-BCL drugs to reduce platelet toxicity. Their compound is effective in several tumor models in vivo and had reduced toxicity in three patients with refractory leukemia.
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Drug Discovery
JOBS of the week
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Careers

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Career snapshots archive
Career snapshots feature people associated with drug discovery and drug development, with the aim of providing expert insights and advice on a wide range of positions and career paths in this field.
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