Friday, October 5, 2012

Drug Discovery@nature.com 5 October 2012

Drug Discovery

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Comparing the Performance of Antibodies Generated From Peptide and DNA-Encoded Antigens
Ross Chambers, PhD, Director, R&D,
Oct 16 at 1pm EST.

A dirty secret of the antibody world is that most antibodies don't work. A large study generated comparative data proving DNA-encoded antigens produce quality antibodies at a much higher success rate than with peptide antigens.
TABLE OF CONTENTS

5 October 2012

News
Analysis
Research Highlights
Research & Reviews
Careers


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ePOSTER ON METABOLIC SYNDROME

Published originally in 2011, the 2012 version of the ePoster features a new organ -- the pancreas -- plus updates for the existing organs to reflect key advances of the past year.

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News

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Economists propose a US$30 billion boost to biomedical R&D
doi:10.1038/nrd3857
Economists hope they can attract billions of dollars for drug R&D by securitizing research projects. Could they close the innovation gap in the process?
Full Text

Moving from an asthma pipe dream to a pipeline
doi:10.1038/nrd3858
After decades of stubbornly slow progress in asthma drug development, recent results from a trial of GlaxoSmithKline's mepolizumab hint at a brighter future.
Full Text

Biobusiness Briefs: Dual-acting combination meets heart failure end point
doi:10.1038/nrd3855
Novartis has announced positive results from the Phase II trial of its first-in-class angiotensin receptor neprilysin inhibitor combination, LCZ696.
Full Text

Market watch: Upcoming market catalysts in Q4 2012
doi:10.1038/nrd3856
Key market catalysts include an expected decision by the FDA on the approval of the anticancer drug cabozantinib; results from a trial of the peptide NX-1207 in benign prostatic hypertrophy; and results from a trial of interferon-free regimens for HCV infection.
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Analysis

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Resetting the clock in diabetes
doi:10.1038/scibx.2012.995
Researchers have evidence that pancreatic islet β cells do not die but rather dedifferentiate in mouse models of type 1 and type 2 diabetes. The findings suggest that reawakening these dormant cells might restore insulin secretion in diabetics.
Full Text

From the analyst's couch: Autism spectrum disorders
doi:10.1038/nrd3771
This analysis looks at the increasing number of candidates in the pipeline for autism spectrum disorders, reflecting the increasing prevalence of autism and the growing interest in finding novel treatments.
Full Text

Research Highlights

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Neurodegenerative diseases: Anti-epileptic drug shows benefit in AD mouse model
doi:10.1038/nrd3850
Using a mouse model engineered to overexpress human amyloid precursor protein and amyloid-β, researchers have shown that cognitive and synaptic deficits are caused by aberrant neuronal network activity, and that this can be improved with an anti-epileptic drug.
Full Text

Vaccines: Self-amplifying RNA in lipid nanoparticles: a next-generation vaccine?
doi:10.1038/nrd3854
A new vaccine platform based on self-amplifying RNA encapsulated in synthetic lipid nanoparticles overcomes some of the limitations of earlier nucleic-acid-based approaches.
Full Text

Metabolic disorders: Safe cannabinoid receptor modulators in sight?
doi:10.1038/nrd3851
A peripherally selective CB1R inverse agonist can safely and effectively reduce body weight in a mouse model of obesity, without affecting behaviour.
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Research & Reviews

Top

Targeting the TGFβ signalling pathway in disease
doi:10.1038/nrd3810
This Review considers why the TGFβ signalling pathway is a drug target, the potential clinical applications of TGFβ inhibition, the issues arising with anti-TGFβ therapy and how these might be tackled.
Full Text

Targeting cells in chronic inflammation
doi:10.1038/nrd3794
This Review focuses on the current knowledge of the IL-17–TH17 cell pathway to better understand the positive as well as potential negative consequences of targeting them.
Full Text

Naratriptan mitigates CGRP1-associated motor neuron degeneration caused by an expanded polyglutamine repeat tract
doi:10.1038/nm.2932
Researchers describe a molecular cascade whereby mutant androgen receptor upregulates CGRP in neuronal cells, promoting JNK activation and degeneration. The 5-HT1B/1D receptor agonist naratriptan decreases CGRP expression and improves motor performance in a mouse model of SBMA.
Full Text

Discovery of an allosteric mechanism for the regulation of HCV NS3 protein function
doi:10.1038/nchembio.1081
Researchers propose that compounds binding a newly discovered allosteric site of the hepatitis C virus’s NS3 protein may inhibit its function, and thus represent a new class of direct-acting antiviral agents.
Full Text

Drug Discovery
JOBS of the week
Postdoctoral Fellow to Study Molecular Mechanisms of Anti-Cancer Drug Resistance
Texas Tech University Health Science Center School of Medicine Cancer Center
Drug Discovery Programme - Head of Biology
Beatson Institute for Cancer Research
Postdoctoral in Chemical Biology for Drug Discovery in Parasitology
GlaxoSmithKline
Postdoctoral Fellowship in Synthetic Cell-Based Screening / Microfluidics / Drug Discovery
The Scripps Research Institute (TSRI)
Post Doctoral Fellowship - Bacterial Pathogenesis and Antimicrobial Drug Discovery
Beth Israel Deacon Medical Center - Harvard Medical School
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Drug Discovery
EVENT
Biosimilar Drug Development World Americas 2012
27.-30.11.12
WA, US
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Careers

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Career snapshots archive
Career snapshots feature people associated with drug discovery and drug development, with the aim of providing expert insights and advice on a wide range of positions and career paths in this field.
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