Friday, May 11, 2012

Drug Discovery@nature.com 11 May 2012

Drug Discovery

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TABLE OF CONTENTS

11 May 2012

News
Analysis
Research Highlights
Research & Reviews
Careers
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News

Top

Drug-making plant blooms
doi:10.1038/485160a
Approval of a 'biologic' manufactured in plant cells may pave the way for similar products.
Full Text

Stromedix acquisition signals growing interest in fibrosis
doi:10.1038/nbt0512-375
A deal in which Biogen Idec purchased the startup Stromedix indicates growing optimism that better biological targets are being identified and addressed in the underserved indication of fibrosis.
Full Text

Deal watch: Alcon invests in first non-surgical therapy for common eye disorder
doi:10.1038/nrd3736
ThromboGenics has entered into a commercialization agreement with Alcon for its experimental therapeutic ocriplasmin, which has successfully completed Phase III trials for an eye disorder known as symptomatic vitreomacular adhesion.
Full Text

Affymax poised to challenge Amgen
doi:10.1038/nbt0512-377
The 20-year dominance of Amgen's erythropoietins in the US anemia market looks like it may be coming to an end.
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Analysis

Top

Heart beats fat
doi:10.1038/scibx.2012.455
The findings that knocking down microRNA-208a in the heart leads to systemic benefits in obesity and metabolic diseases could expand the potential indications for miRagen's antimiR-208, which is in preclinical development for cardiac hypertrophy.
Full Text

Fresh from the Pipeline: Ivacaftor
doi:10.1038/nrd3723
First disease-modifying drug approved in the United States for the treatment of cystic fibrosis in patients with a specific mutation in the gene encoding the cystic fibrosis transmembrane conductance regulator.
Full Text

From the analyst's couch: Drug development risk and the cost of capital
doi:10.1038/nrd3722
This article analyses the relationship between risk and the cost of capital for projects in different stages of drug development and describes a framework that could improve portfolio optimization strategies.
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Research Highlights

Top

Neurodegenerative disease: The stress of misfolding
doi:10.1038/nrd3731
Two studies provide evidence that α-synuclein-induced endoplasmic reticulum (ER) stress has a crucial role in promoting neurodegeneration in α-synucleinopathies, and that targeting chronic ER stress may represent a plausible target for future therapies.
Full Text

Cancer genomics: Constructing a 'cancerpaedia'
doi:10.1038/nrd3730
Two recent papers published in Nature report on genomic changes in cancer cell lines that indicate sensitivity to targeted drugs.
Full Text

Mouse models: Of mice and men
doi:10.1038/nrc3270
A clinical trial in mice with lung cancer indicates the likely efficacy of the MEK inhibitor selumetinib in a current ongoing human clinical trial.
Full Text

Research & Reviews

Top

Epigenetic protein families: a new frontier for drug discovery
doi:10.1038/nrd3674
In this article, the authors review the protein families that mediate epigenetic signalling through histone acetylation and methylation, and highlight progress in the pharmacological modulation of each class of proteins.
Full Text

Intra-tumour heterogeneity: a looking glass for cancer?
doi:10.1038/nrc3261
This Review outlines both genetic and non-genetic causes of phenotypic heterogeneity of tumour cells and the implications of intra-tumour heterogeneity in diagnostics and the development of therapeutic resistance.
Full Text

The deubiquitinase USP9X suppresses pancreatic ductal adenocarcinoma
doi:10.1038/nature11114
A transposon-mediated insertional mutagenesis screen reveals inactivation of the X-linked deubiquitinase gene Usp9x in over 50% of pancreatic ductal adenocarcinomas, suggesting Usp9x has prognostic and therapeutic relevance for this disease.
Full Text

A selective inhibitor reveals PI3Kγ dependence of TH17 cell differentiation
doi:10.1038/nchembio.957
A chemoproteomic approach adapted for high-throughput screening leads to the identification of a selective PI3Kγ inhibitor. Application of this inhibitor in human and mouse cellular models reinforces selective inhibition of PI3Kγ as a potential treatment for inflammatory and autoimmune diseases.
Full Text

Drug Discovery
JOBS of the week
PhD student for Biomedical Imaging Group Rotterdam (BIGR) - on the project Imaging biomarkers for oncology drug development
Erasmus MC
Post-doc 'The development of novel antibody drug conjugates'
VU University Medical Center
Drug Safety Operations Manager - Permanent Job
Yoh
Drug Saftey Coordinator Job
Yoh
Observational, prospective study about the incidence of adverse drug effects in patients with drug-resistence epilepsy
Università degli Studi di Firenze- Dipartimento di Scienze Neurologiche e Psichiatriche
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Drug Discovery
EVENT
DDI and ETS-2012: 15th international Drug-Drug Interaction and 10th Early Toxicity Screening conferences
11.-15.06.12
WA, US
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Careers

Top

Career snapshots archive
Career snapshots feature people associated with drug discovery and drug development, with the aim of providing expert insights and advice on a wide range of positions and career paths in this field.
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